Lebitso | Cetrorelix acetate |
Nomoro ea CAS | 120287-85-6 |
Mokhoa oa limolek'hule | Setšoantšo sa C70H92ClN17O14 |
Boima ba molek'hule | 1431.04 |
Nomoro ea EINECS | 686-384-6 |
AC-(D-ALA[3-(2-NAPHTHYL)])-[D-PHE(4-CL)]-(D-ALA[3-(3-PYRIDYL)])-SER-TYR-(D-CIT)-LEU-ARG-PRO-D-ALA-OH;Cetrorelixacetate;CETRORELIHLOHLOKO;CETRORELIHLOKO;CETRORELIHLOM;CETRORELIX;CETRICEDRICETRIXEDRICEDRIXEDRIXEDRIXRIX; hemicalbookN-Acetyl-3-(2-naphthalenyl)-D-Ala-4-chloro-D-Phe-3-(3-pyridyl)-D-Ala-L-Ser-L-Tyr-N5-(aminocarbonyl)-D-Orn-L-Leu-L-Arg-L-Pro-D-Cem2;Ala-Troli-Pro-D-Cem.
Cetrorelix acetate ke decapeptide ea maiketsetso, e sebelisoang haholo theknoloji e thusang ho ba le bana ho thibela ho hlaha ha mahe pele ho nako ho bakuli ba nang le ts'usumetso e laoloang ea mahe a bomme. Ke mohanyetsi oa gonadotropin-release hormone (GnRH) ea ka qothisanang lehlokoa le LHRH e sa feleng ho tlama li-receptor tse ka har'a lera la sele ea pituitary, ka tsela eo e thibela secretion ea luteinizing hormone (LH) le follicle stimulating hormone (FSH) ke pituitary ka mokhoa o itšetlehileng ka tekanyo.
Cetrorelix acetate ke mohanyetsi oa gonadotropin-releasing hormone (GnRH). Sehlahisoa sena se qothisana lehlokoa le GnRH ea endogenous bakeng sa li-receptor tsa lisele tsa pituitary, ka tsela eo e thibela ho lokolloa ha hormone ea "luteinizing" (LH) le follicle-stimulating hormone (FSH), e liehisa ponahalo ea LH, ka tsela eo e laola ho ruruha. Phello ea sehlahisoa sena e itšetlehile ka tekanyo ea tekanyo, phello ea inhibitory e tobileng, 'me e bolokoa ke phekolo e tsoelang pele, ntle le ho baka keketseho ea pele ea mosebetsi oa progesterone receptor e lateloa ke ho fokotseha.
Bate ea metsi ea tšepe ea thermostatic ea motlakase
Sebōpi sa ho hanyetsa mofuta oa lebokose
Motlakase o futhumatsang mocheso o sa khaotseng oa onto ea ho omisa
Li-incubators tse futhumetseng
Insoluble particle analyzer
Chromatography ea metsi
Polarimeter e ikemetseng
spectrometer ea infrared
UV / Photometer e bonahalang
Lebokose la ho omisa lebokoso la ho futhumatsa la motlakase
Sterilizer e otlolohileng ea khatello ea mouoane
PH mitha
Hlakola Tester
Teko ea Osmolality
Khasete Mongobo Analyzer
Multi-parameter analyzer
Lebokose la ho omisa la motlakase
Biochemical incubator
Seqhoala sa hlobo
Aseptic isolator
Kakaretso ea organic carbon detector
Setsi sa Vacuum sa Desktop
Comprehensive drug stability test chamber
Sinki ea kamehla ea mocheso le ho hlapa metsi
Lebokose la polokelo la sehatsetsing sa bongaka
Chromatograph ea Khase
Khabinete ea polokeho ea baeloji
Benche e hloekileng
TOC le conductivity ea phepelo ea mantlha le lintlha tsa ho khutlisa li hlahlojoa nako le nako. TOC e behiloe leihlo ke QC beke e 'ngoe le e 'ngoe. Conductivity e beoa leihlo inthaneteng 'me e rekotoa ke opareitara ea seteishene sa metsi a hloekisitsoeng hang ka mor'a lihora tse ling le tse ling tse nne. The conductivity e hlahlojoa ho RO ea mantlha, RO ea bobeli, EDI le kakaretso ea ho khutlisa mokhoa oa ho tsamaisa. Litlhaloso tsa metsi a hloekisitsoeng li teng 'me li lumellana le litlhaloso tse boletsoeng esale pele tse sa feteng 1.3 µs/cm ho 25°C (USP). Bakeng sa phepelo ea mantlha le lintlha tsa ho khutla, tlhahlobo e felletseng. e etsoa beke e 'ngoe le e 'ngoe, bakeng sa lintlha tse ling tse sebelisoang ho lupu e potolohang, tlhahlobo e felletseng e etsoa hang ka khoeli. Teko e felletseng e kenyelletsa litlhaku, pH, nitrate, nitrite, ammonia, conductivity, TOC, lintho tse sa fetoheng, lirafshoa tse boima, meeli ea likokoana-hloko le endotoxin ea baktheria.