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Semaglutide bakeng sa Mofuta oa 2 oa lefu la tsoekere

Tlhaloso e Khutšoanyane:

Lebitso: Semaglutide

Nomoro ea CAS: 910463-68-2

Mokhoa oa molek'hule: C187H291N45O59

Boima ba molek'hule: 4113.57754

Nomoro ea EINECS: 203-405-2


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Lintlha tsa Sehlahisoa

Lebitso Semaglutide
Nomoro ea CAS 910463-68-2
Mokhoa oa limolek'hule C187H291N45O59
Boima ba molek'hule 4113.57754
Nomoro ea EINECS 203-405-2

Litlhaloso tse tšoanang

Sermaglutide;Semaglutide fandachem;ho se hloeke ha Semaglutide;Sermaglutide USP / EP;semaglutide;Sermaglutide CAS 910463 68 2;Ozempic,

Tlhaloso

Semaglutide ke moloko o mocha oa li-analogues tsa GLP-1 (glucagon-like peptide-1), 'me semaglutide ke mofuta oa litekanyetso tse nkang nako e telele o thehiloeng ho latela sebopeho sa mantlha sa liraglutide, se nang le phello e betere kalafong ea lefu la tsoekere la mofuta oa 2.Novo Nordisk e phethile lithuto tsa 6 Phase IIIa ea ente ea semaglutide, 'me e rometse kopo e ncha ea ho ngolisa lithethefatsi bakeng sa ente ea beke le beke ea semaglutide ho US Food and Drug Administration (FDA) ka December 5, 2016. Kopo ea Phatlalatso ea Khoebo (MAA) e boetse e romelloa ho European Medicines Agency (EMA).

Ha e bapisoa le liraglutide, semaglutide e na le ketane e telele ea aliphatic le ho eketseha ha hydrophobicity, empa semaglutide e fetotsoe ka ketane e khutšoanyane ea PEG, 'me hydrophilicity ea eona e ntlafatsoa haholo.Ka mor'a phetoho ea PEG, e ke ke ea tlama haufi-ufi feela le albumin, e koahela sebaka sa enzymatic hydrolysis ea DPP-4, empa hape e fokotsa ho tsoa ha renal, ho lelefatsa halofo ea bophelo, le ho finyella phello ea nako e telele ea ho potoloha.

Kopo

Semaglutide ke mofuta oa litekanyetso tsa nako e telele o ntlafalitsoeng ho latela sebopeho sa mantlha sa liraglutide, se sebetsang hantle ho alafa lefu la tsoekere la mofuta oa 2.

Bioactivity

Semaglutide (Rybelsus, Ozempic, NN9535, OG217SC, NNC0113-0217) ke analogue ea nako e telele ea glucagon-joaloka peptide 1 (GLP-1), agonist ea GLP-1receptor, e nang le mofuta oa 2 oa Phekolo e sebetsang hantle ea lefu la tsoekere (TDM diabetes mellitus). ).

Tsamaiso ea Boleng

Ka kakaretso, tsamaiso ea boleng le tiisetso li teng ho akaretsa mekhahlelo eohle ea tlhahiso ea sehlahisoa se felileng.Ts'ebetso e lekaneng ea tlhahiso le taolo e etsoa ho latela mekhoa / litlhaloso tse amohetsoeng.Taolo ea phetoho le tsamaiso ea ho kheloha e teng, 'me ho ile ha etsoa tlhahlobo le lipatlisiso tse hlokahalang.Mekhoa e nepahetseng e teng ho netefatsa boleng ba sehlahisoa pele se lokolloa 'marakeng.


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