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Tianeptine bakeng sa sistimi ea 5-HT, sedation, anti-anti-actylcholine le pelo ea pelo bakeng sa khatello ea maikutlo

Tlhaloso e khutšoane:

Lebitso la Senyesemane: Tianeptine sulfate

Nomoro ea Cas: 1224690-94-9

Foromo ea limolecular: C42h56cl2n4o14s3

Boima ba moleng: 1008.013444


Lintlha tsa sehlahisoa

Li-tag tsa lihlahisoa

Lintlha tsa sehlahisoa

Lebitso Tianeptine
Nomoro ea CAS 1224690-84-9
Foromo ea limolecular C21h27cln2o8s2
Boima ba Molecular 535.02
Ntlha ea ho qhibiliha 129-131 ° C
Poleft Point 609.2ºC ho 760 mmhg
Bohloeki 99%
Polokelo E tiisitsoeng ka mocheso o omileng, oa kamore ea kamore
Foromo Phofo
Mmala Tšoeu
Packing Pla ea mokotla + aluminium Bag

Synonyms

Thm; Tianepneyhydrate Der / Tianeptinulfte

Phello ea pharmaColoCologana

Phello ea pharmaColoCologana

1. Mokhoa oa antidestant oa sehlahisoa sena o fapane le oa setso sa tca. E ka eketsa ho nyoloha ha 5-HT ho Conaptic Cleft ea Synaptic, empa e na le phello e fokolang ho buuptake ea 5-Ht le na. E kanna ea ba le phello ea ho ntlafatsa phetisetso ea 5-ht. Ha e na khethollo bakeng sa li-receptors, H1, α1 le α2-na basetlelete.
2. Ho sebetsa hantle ha sehlahisoa sena ho tšoana le tsa TCA, 'me polokeho ea eona e molemo ho feta TCA (li-antisepress tsa eona tse ntle). Ho sebetsa hantle ha sehlahisoa sena ho tšoana le sa SSR Cluototine.
3. Liteko tsa lithethefatsi li bontšitse hore li ka re: Eketsa tšebetso e itlhahelang feela ea lisele tsa pyramidal ka ho hlaphoheloa tšebetsong ea eona kamora ts'ebetso ea eona ka mor'a ho tlohela mosebetsi. Eketsa ho nchafatsa ha hydroustyptory ea 5-hydroxyttryptomine ea li-neuron Cortex le hippocampus.

 

Lipatlisiso tsa TOXCOPology

- Ho hlobaela ka thata le liteko tsa nako e telele: Ha ho liphetoho tse telele: ha ho liphetoho ho biology, sebetsa ka sebete, thuto ea patrophone.
- Tlhahlobo ea chefo: TAINEPTINE ha e na tšusumetso ho bokhoni ba batsoali ba tšoaroang hammoho le masedun le bana.
- Teko ea mutaven: Tianeptine ha e na matla a holimo.

 

Litlamorao

- Bohloko ba epiland, ho bohloko ba ka mpeng, molomo o omileng, ho iphahamisang, ho nyefola, ho hlatsa, ho soma ha pelo;
- Ho hloka boroko, ho otsela, litoro tsa bosiu, bofokoli;
- Tachycardia, tse ikhethang, bohloko ba pelehi;
- Ho khopisisa, hlooho ea hlooho, ea hlohlelletsang, ho thothomela ha sefahleho;
- Ho hema hanyane ka ho hema, maikutlo a ho sithabela 'metso;
- imalgia, bohloko ba morao, jj.


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  • E 'ngoe:

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