Ho khomarela tumelo ea "Ho theha lintho tsa maemo a holimo le ho theha metsoalle le batho kajeno ba tsoang lefats'eng lohle", re tloaetse ho beha thahasello ea bareki sebakeng sa pele bakeng sa theko e qotsitsoeng bakeng sa China Healthy Weight Loss CAS 96829-58-2 99% Bulk API Rimonbant CetilistatOrlistat, Ho tloha ha ho thehoa ka hare ho lilemo tsa pele tsa 1990, re se re hahile marang-rang a rona a thekiso USA, Jeremane, Asia, le linaheng tse 'maloa tsa Bochabela bo Hare. Re ikemiselitse ho fumana morekisi oa maemo a holimo bakeng sa OEM lefatšeng ka bophara le ka morao-rao!
Ka ho tšoarella tumelong ea "Ho theha lintho tsa maemo a holimo le ho theha metsoalle le batho ba tsoang lefats'eng lohle kajeno", re tloaetse ho beha lithahasello tsa bareki sebakeng sa pele bakeng saChina 96829-58-2, Orlistat, Ka tsamaiso ea morao-rao e phethahetseng ea ho fana ka maikutlo a ho bapatsa le mosebetsi o boima oa basebetsi ba 300 ba nang le litsebo, k'hamphani ea rona e ntlafalitse mefuta eohle ea tharollo ho tloha boemong bo phahameng, ba maemo a mahareng ho isa boemong bo tlaase. Khetho ena eohle ea lintho tse ntle e fa bareki ba rona likhetho tse fapaneng. Ntle ho moo, k'hamphani ea rona e khomarela boleng ba boleng bo holimo le theko e utloahalang, hape re u fa litšebeletso tse ntle tsa OEM ho lihlahisoa tse ngata tse tummeng.
| Lebitso | Leuprorelin |
| Nomoro ea CAS | 53714-56-0 |
| Mokhoa oa limolek'hule | Setšoantšo sa C59H84N16O12 |
| Boima ba molek'hule | 1209.4 |
| Nomoro ea EINECS | 633-395-9 |
| Ho potoloha ho itseng | D25 -31.7° (c = 1 ho 1% acetic acid) |
| Botenya | 1.44±0.1 g/cm3(E boletsoeng esale pele) |
| Boemo ba polokelo | -15°C |
| Sebopeho | E makhethe |
| Acidity coefficient | (pKa) 9.82±0.15 (E boletsoeng esale pele) |
| Ho qhibiliha ha metsi | E qhibiliha ka metsing ka 1mg/ml |
LH-RHLEUPROLIDE;LEUPROLIDE;LEUPROLIDE(HUMAN);LEUPRORELIN;[DES-GLY10,D-LEU6,PRO-NHET9]-LUTEINIZINGHORMONE-RELEASINGHORMONEHUMAN;(DES-GLY10,D-LEU6,PRO -NHET9)-LUTEINIZINGHORMONE-RELEASINGHORMONE;(DES-GLY10,D-LEU6,PRO-NHET9)-LUTEINIZINGHORMONE-RELEASINGFACTOR;[DES-GLY10,D-LEU6,PRO-NHET9]-LH-RH(BATHO)
Leuprolide, goserelin, triprelin, le nafarelin ke litlhare tse 'maloa tse sebelisoang hangata litsing tsa bongaka ho tlosa mae a bomme bakeng sa kalafo ea mofets'e oa pele ho nako le mofets'e oa senya. (e bitsoang lithethefatsi tsa GnRH-a), lithethefatsi tsa GnRH-a li tšoana ka sebopeho le GnRH 'me li hlōlisana le li-receptor tsa pituitary GnRH. Ke hore, gonadotropin e hlahisoang ke pituitary e fokotseha, e lebisang ho fokotseha ho hoholo ha hormone ea thobalano e hlahisoang ke ovary.
Leuprolide ke analoge ea gonadotropin-release hormone (GnRH), peptide e entsoeng ka li-amino acid tse 9. Sehlahisoa sena se ka thibela ka katleho mosebetsi oa tsamaiso ea pituitary-gonadal, ho hanyetsa li-enzyme tsa proteolytic le kamano ea pituitary receptor ea GnRH e matla ho feta GnRH, 'me mosebetsi oa ho khothalletsa ho lokolloa ha hormone ea luteinizing (LH) e ka bang makhetlo a 20 a GnRH. E boetse e na le phello e matla ea inhibitory mosebetsing oa pituitary-gonad ho feta GnRH. Mothating oa pele oa kalafo, follicle stimulating hormone (FSH), LH, estrogen kapa androgen e ka eketseha ka nakoana, ebe, ka lebaka la ho fokotseha ha karabelo ea tšoelesa ea pituitary, secretion ea FSH, LH le estrogen kapa androgen e thibetsoe, e bakang ho itšetleha ka lihomone tsa thobalano. Mafu a thobalano (a kang kankere ea prostate, endometriosis, joalo-joalo) a na le phello ea phekolo.
Hajoale, letsoai la acetate la leuprolide le sebelisoa haholo ka bongaka, hobane ts'ebetso ea leuprolide acetate e tsitsitse haholoanyane mocheso oa kamore. Mokelikeli o lokela ho lahloa. E ka sebelisoa bakeng sa kalafo castration lithethefatsi endometriosis le uterine fibroids, bohareng precocious puberty, premenopausal kankere ea matsoele le kankere ea tšoelesa ea senya, 'me hape bakeng sa tshebetso uterine tsoa mali e contraindicated kapa e sa sebetseng bakeng sa phekolo e tloaelehileng ea hormone. E ka boela ea sebelisoa e le premedication pele endometrial resection, e ka ka tsela e leka-lekaneng ho tšesa endometrium, ho fokotsa edema, le ho fokotsa bothata ba ho buuoa.Ho khomarela tumelo ea "Ho theha lintho tse phahameng ka ho fetisisa le ho theha metsoalle le batho ba kajeno ba tsoang lefats'eng lohle", re atisa ho beha thahasello ea bareki sebakeng sa pele bakeng sa Theko e qotsitsoeng bakeng sa China Healthy Weight 92 Los 92 Los 92 Los 92 Los 92 Los API Rimonbant Cetilistat Orlistat, Ho tloha ha e thehoa ka hare ho 1990s ea pele, re se re hahile marang-rang a rona a thekiso USA, Jeremane, Asia le linaheng tse 'maloa tsa Bochabela bo Hare. Re ikemiselitse ho fumana morekisi oa maemo a holimo bakeng sa OEM lefatšeng ka bophara le ka morao-rao!
Theko e qotsitsoeng bakeng saChina 96829-58-2, Orlistat, Ka mokhoa oa morao-rao oa ho fana ka maikutlo a ho bapatsa ka mokhoa o phethahetseng le mosebetsi o boima oa basebetsi ba 300 ba nang le tsebo, k'hamphani ea rona e hlahisitse mefuta eohle ea tharollo ho tloha boemong bo phahameng, ba maemo a mahareng ho isa boemong bo tlaase. Khetho ena eohle ea lintho tse ntle e fa bareki ba rona likhetho tse fapaneng. Ntle ho moo, k'hamphani ea rona e khomarela boleng ba boleng bo holimo le theko e utloahalang, hape re u fa litšebeletso tse ntle tsa OEM ho lihlahisoa tse ngata tse tummeng.