tsoela pele ho ntlafatsa, ho ba le tharollo e itseng ea boleng bo holimo ho ipapisitse le litlhoko tsa maemo a mmaraka le tsa bareki. Mokhatlo oa rona o na le lenaneo le letle la netefatso le thehiloe bakeng sa PriceList bakeng sa Phano ea Factory ea boleng bo holimo ea China.OrlistatPowder CAS 96829-58-2, "Boleng", "botšepehi" le "tšebeletso" ke molao-motheo oa rona. Botšepehi ba rona le boitlamo ba rona bo lula ka tlhompho ho mofani oa hau. Ikopanye le Rona Kajeno Bakeng sa lintlha tse ling, ikopanye le rona hona joale.
tsoela pele ho ntlafatsa, ho ba le tharollo e itseng ea boleng bo holimo ho ipapisitse le litlhoko tsa maemo a mmaraka le tsa bareki. Mokhatlo oa rona o na le lenaneo le letle la netefatso le thehiloe bakeng saChina Orlistat phofo, Orlistat, Re lumela hore ka ts'ebeletso ea rona e tsoileng matsoho u ka fumana ts'ebetso e ntle ka ho fetesisa le ho bitsa lihlahisoa tse tlase ho rona ka nako e telele. Re itlama ho fana ka litšebeletso tse betere le ho etsa boleng bo eketsehileng ho bareki bohle ba rona. Re tšepa hore re ka theha bokamoso bo molemo hammoho.
| Lebitso | Leuprorelin |
| Nomoro ea CAS | 53714-56-0 |
| Mokhoa oa limolek'hule | Setšoantšo sa C59H84N16O12 |
| Boima ba molek'hule | 1209.4 |
| Nomoro ea EINECS | 633-395-9 |
| Ho potoloha ho itseng | D25 -31.7° (c = 1 ho 1% acetic acid) |
| Botenya | 1.44±0.1 g/cm3(E boletsoeng esale pele) |
| Boemo ba polokelo | -15°C |
| Sebopeho | E makhethe |
| Acidity coefficient | (pKa) 9.82±0.15 (E boletsoeng esale pele) |
| Ho qhibiliha ha metsi | E qhibiliha ka metsing ka 1mg/ml |
LH-RHLEUPROLIDE;LEUPROLIDE;LEUPROLIDE(HUMAN);LEUPRORELIN;[DES-GLY10,D-LEU6,PRO-NHET9]-LUTEINIZINGHORMONE-RELEASINGHORMONEHUMAN;(DES-GLY10,D-LEU6,PRO -NHET9)-LUTEINIZINGHORMONE-RELEASINGHORMONE;(DES-GLY10,D-LEU6,PRO-NHET9)-LUTEINIZINGHORMONE-RELEASINGFACTOR;[DES-GLY10,D-LEU6,PRO-NHET9]-LH-RH(BATHO)
Leuprolide, goserelin, triprelin, le nafarelin ke litlhare tse 'maloa tse sebelisoang hangata litsing tsa bongaka ho tlosa mae a bomme bakeng sa kalafo ea mofets'e oa pele ho nako le mofets'e oa senya. (e bitsoang lithethefatsi tsa GnRH-a), lithethefatsi tsa GnRH-a li tšoana ka sebopeho le GnRH 'me li hlōlisana le li-receptor tsa pituitary GnRH. Ke hore, gonadotropin e hlahisoang ke pituitary e fokotseha, e lebisang ho fokotseha ho hoholo ha hormone ea thobalano e hlahisoang ke ovary.
Leuprolide ke analoge ea gonadotropin-release hormone (GnRH), peptide e entsoeng ka li-amino acid tse 9. Sehlahisoa sena se ka thibela ka katleho mosebetsi oa tsamaiso ea pituitary-gonadal, ho hanyetsa li-enzyme tsa proteolytic le kamano ea pituitary receptor ea GnRH e matla ho feta GnRH, 'me mosebetsi oa ho khothalletsa ho lokolloa ha hormone ea luteinizing (LH) e ka bang makhetlo a 20 a GnRH. E boetse e na le phello e matla ea inhibitory mosebetsing oa pituitary-gonad ho feta GnRH. Mothating oa pele oa kalafo, follicle stimulating hormone (FSH), LH, estrogen kapa androgen e ka eketseha ka nakoana, ebe, ka lebaka la ho fokotseha ha karabelo ea tšoelesa ea pituitary, secretion ea FSH, LH le estrogen kapa androgen e thibetsoe, e bakang ho itšetleha ka lihomone tsa thobalano. Mafu a thobalano (a kang kankere ea prostate, endometriosis, joalo-joalo) a na le phello ea phekolo.
Hajoale, letsoai la acetate la leuprolide le sebelisoa haholo ka bongaka, hobane ts'ebetso ea leuprolide acetate e tsitsitse haholoanyane mocheso oa kamore. Mokelikeli o lokela ho lahloa. E ka sebelisoa bakeng sa kalafo castration lithethefatsi endometriosis le uterine fibroids, bohareng precocious puberty, premenopausal kankere ea matsoele le kankere ea tšoelesa ea senya, 'me hape bakeng sa tshebetso uterine tsoa mali e contraindicated kapa e sa sebetseng bakeng sa phekolo e tloaelehileng ea hormone. E ka boela ea sebelisoa e le premedication pele endometrial resection, e ka evenly tšesaane endometrium, fokotsa edema, 'me fokotsa bothata ba ho buuoa.tsoela pele ho ntlafatsa, ho ba itseng tharollo boleng bo holimo tumellanong le maraka le moreki ditlhoko maemo a. Mokhatlo oa rona o na le lenaneo le letle la netefatso le thehiloe bakeng sa PriceList bakeng sa China High Quality Factory Supply Orlistat Powder CAS 96829-58-2, "Quality", "botšepehi" le "ts'ebeletso" ke molao-motheo oa rona. Botšepehi ba rona le boitlamo ba rona bo lula ka tlhompho ho mofani oa hau. Ikopanye le Rona Kajeno Bakeng sa lintlha tse ling, ikopanye le rona hona joale.
PriceList bakeng saChina Orlistat phofo, Orlistat, Re lumela hore ka ts'ebeletso ea rona e ntle haholo o ka fumana ts'ebetso e ntle ka ho fetisisa mme o bitsa lihlahisoa tse nyane ho tsoa ho rona nako e telele. Re itlama ho fana ka litšebeletso tse betere le ho etsa boleng bo eketsehileng ho bareki bohle ba rona. Re tšepa hore re ka theha bokamoso bo molemo hammoho.