Melanotan IIke analoge ea maiketsetso ea cyclic heptapeptide eaα-melanocyte-stimulating hormone (α-MSH), ntshetswa pele hotsosa melanogenesis, ntlafatsaTšireletso ea UV, le ho fetolamesebetsi ea thobalano le metabolism. E sebetsa joalo ka aagonist e sa kgethengli-receptor tsa melanocortin, haholo-holoMC1R, MC3R, leMC4R.
Qalong o ile a ithuta bakeng sa eonaho suha matlalolephotoprotectivethepa, Melanotan II e boetse e bontšitse liphello hontlafatso ea libido, takatso ea lijo, letekanyo ea matla, ho etsa hore e be peptide ea lipatlisiso tse ngata tse nang le thahasello ho dermatology, endocrinology, le meriana ea thobalano.
Melanotan II e sebetsa ka ho kenya li-receptor tse 'maloa tsa melanocortin:
MC1R: Lia susumetsatlhahiso ea melanin→ e eketsa mebala ea letlalo le tšireletso ea UV
MC3R / MC4R: Ke karoloho laola takatso ea lijo, ntlafatso ea libido, lematla a homeostasis
E tšela mokoallo oa mali bokong, e susumetsang litsela tse bohareng tsa neurohormonal
Le hoja e sa amoheleha bakeng sa tšebeliso ea meriana, Melanotan II e ithutoa haholo bakeng sa tse latelang:
Phatlalatsotlhahiso ea eumelanin, e isang hoho suoa ha tlhaho
E fana kaliphello tse sireletsang lifotontle le ho ba letsatsing
Monyetla oa ho fokotsa kotsi ea mofetše oa letlalo ho batho ba nang le letlalo le letle
Bontša hoeketsa libido le takatso ea thobalanoho banna le basadi
E rutiloe e le phekolo e ka bang teng bakeng saho se sebetse hantle ha erectile (ED)ka ts'ebetso ea MC4R
Mots'eanongfokotsa takatso ea lijo le ho ja lijoka ho sebetsa ka litsela tsa hypothalamic
Motlatsi o ka bang tenglipatlisiso tsa botenya
Bohloeki bo phahameng ≥ 99%(HPLC & LC-MS e tiisitsoe)
Synthesized kasolid-phase peptide synthesis (SPPS)
Endotoxin e tlase, li-solvents tse setseng tse tlase
E fumaneha kaR&D ho isa tekanyong ea khoebo