• hlooho_banner_01

Melanotan II

Tlhaloso e Khutšoanyane:

Likarolo tsa API:
Bohloeki bo phahameng ≥ 99%
E entsoe ka solid-phase peptide synthesis (SPPS)
Endotoxin e tlase, li-solvents tse setseng tse tlase
E fumaneha ka R&D ho isa boemong ba khoebo


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Melanotan II API

Melanotan IIke analoge ea maiketsetso ea cyclic heptapeptide eaα-melanocyte-stimulating hormone (α-MSH), ntshetswa pele hotsosa melanogenesis, ntlafatsaTšireletso ea UV, le ho fetolamesebetsi ea thobalano le metabolism. E sebetsa joalo ka aagonist e sa kgethengli-receptor tsa melanocortin, haholo-holoMC1R, MC3R, leMC4R.

Qalong o ile a ithuta bakeng sa eonaho suha matlalolephotoprotectivethepa, Melanotan II e boetse e bontšitse liphello hontlafatso ea libido, takatso ea lijo, letekanyo ea matla, ho etsa hore e be peptide ea lipatlisiso tse ngata tse nang le thahasello ho dermatology, endocrinology, le meriana ea thobalano.


Mokhoa oa Ts'ebetso

Melanotan II e sebetsa ka ho kenya li-receptor tse 'maloa tsa melanocortin:

  • MC1R: Lia susumetsatlhahiso ea melanin→ e eketsa mebala ea letlalo le tšireletso ea UV

  • MC3R / MC4R: Ke karoloho laola takatso ea lijo, ntlafatso ea libido, lematla a homeostasis

  • E tšela mokoallo oa mali bokong, e susumetsang litsela tse bohareng tsa neurohormonal


Lipatlisiso le Likopo tse ka Etsisoang

Le hoja e sa amoheleha bakeng sa tšebeliso ea meriana, Melanotan II e ithutoa haholo bakeng sa tse latelang:

1. Letlalo la Pigmentation & Tšireletso ea UV

  • Phatlalatsotlhahiso ea eumelanin, e isang hoho suoa ha tlhaho

  • E fana kaliphello tse sireletsang lifotontle le ho ba letsatsing

  • Monyetla oa ho fokotsa kotsi ea mofetše oa letlalo ho batho ba nang le letlalo le letle

2. Bothata ba ho Kopanela Liphate

  • Bontša hoeketsa libido le takatso ea thobalanoho banna le basadi

  • E rutiloe e le phekolo e ka bang teng bakeng saho se sebetse hantle ha erectile (ED)ka ts'ebetso ea MC4R

3. Takatso le Boima ba Boima

  • Mots'eanongfokotsa takatso ea lijo le ho ja lijoka ho sebetsa ka litsela tsa hypothalamic

  • Motlatsi o ka bang tenglipatlisiso tsa botenya


API Features (ka Gentolex Group)

  • Bohloeki bo phahameng ≥ 99%(HPLC & LC-MS e tiisitsoe)

  • Synthesized kasolid-phase peptide synthesis (SPPS)

  • Endotoxin e tlase, li-solvents tse setseng tse tlase

  • E fumaneha kaR&D ho isa tekanyong ea khoebo


  • E fetileng:
  • E 'ngoe:

  • Ngola molaetsa wa hao mona mme o re romele wona