Melanotan 1ke analoge ea maiketsetso ea peptide eaα-MSH (hormone e susumetsang ea alpha-melanocyte). E sebetsa kaho kenya tšebetsong melanocortin-1 receptors (MC1R)ho susumetsatlhahiso ea melanin, ho fana ka tlhaholetlalo la mmalaletšireletso ea lifoto.
E bilee amohelehang bakeng sa phekolo ea erythropoietic protoporphyria (EPP)-bothata bo sa tloaelehang bo bakang kutlo e feteletseng ea khanya ea letsatsi. Melanotan 1 e thusa ho eketsehaho mamella mabone a UV, fokotsaliketso tsa phototoxic, le ho ntlafatsatšireletso ea letlalo khahlanong le tšenyo e bakoang ke UV.
KhethangMC1R agonist
Ea eketsehatlhahiso ea eumelanin
E fana katshireletso letsatsing la tlhaho
TšehetsaTokiso ea DNA le karabelo e khahlanong le ho ruruha
Monyetla bakeng savitiligo, thibelo ea mofetše oa letlalo, lecosmetic pigmentation
E hlahlobiloe ka har'athibela botsofalilephekolo ea dermatological
Bohloeki bo phahameng ≥99%
Solid-phase peptide synthesis (SPPS)
Litekanyetso tsa tlhahiso tse kang GMP
Phepelo e ka fokotsoang: R&D ho isa maemong a khoebo